Search results for " bromide"

showing 10 items of 315 documents

Deprotonation of Benzoxazole and Oxazole Using Lithium Magnesates

2005

International audience; The first deprotonations of oxazole and benzoxazole using lithium magnesates are described. The reactions occurred in tetrahydrofuran at room temperature using 1/3 equiv of lithium tributylmagnesate. As 2-lithiooxazole and 2-lithiobenzoxazole, lithium tri(2-oxazolyl)magnesate and lithium tri(2-benzoxazolyl)magnesate very rapidly and completely isomerized to the more stable 2-(isocyano)enolate and 2-(isocyano)phenolate type structures, respectively, a result shown by NMR analysis. The isolation of 2-substituted oxazoles and benzoxazoles in medium to good yields after electrophilic trapping was interpreted in two ways:  (1) the equilibration between the open and closed…

010405 organic chemistryLithium bromide[CHIM.ORGA]Chemical Sciences/Organic chemistryOrganic Chemistrychemistry.chemical_element[CHIM.THER]Chemical Sciences/Medicinal Chemistry[CHIM.MATE]Chemical Sciences/Material chemistry[CHIM.CATA]Chemical Sciences/CatalysisBenzoxazole[CHIM.INOR]Chemical Sciences/Inorganic chemistry010402 general chemistryPhotochemistry01 natural sciencesMedicinal chemistry0104 chemical scienceschemistry.chemical_compoundDeprotonationchemistryIntramolecular forceElectrophile[CHIM]Chemical SciencesLithium[CHIM.RADIO]Chemical Sciences/RadiochemistryTetrahydrofuranOxazole
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Indicaxanthin from Opuntia Ficus Indica (L. Mill) impairs melanoma cell proliferation, invasiveness, and tumor progression.

2018

Abstract Background: A strong, reciprocal crosstalk between inflammation and melanoma has rigorously been demonstrated in recent years, showing how crucial is a pro-inflammatory microenvironment to drive therapy resistance and metastasis. Purpose: We investigated on the effects of Indicaxanthin, a novel, anti-inflammatory and bioavailable phytochemical from Opuntia Ficus Indica fruits, against human melanoma both in vitro and in vivo. Study Design and Methods: The effects of indicaxanthin were evaluated against the proliferation of A375 human melanoma cell line and in a mice model of cutaneous melanoma. Cell proliferation was assessed by MTT assay, apoptosis by Annexin V-Fluorescein Isothio…

0301 basic medicine3003MaleSkin NeoplasmsPyridinesPyridinePhytochemicalsMelanoma ExperimentalPharmaceutical ScienceIndicaxanthinApoptosisBcl-2 B cell lymphoma gene-2 (Bcl-2)chemistry.chemical_compoundMice0302 clinical medicineOpuntia Ficus Indica (L.Mill)Settore BIO/10 - BiochimicaDrug DiscoveryCXCL1 chemokine (C-X-C motif) ligand 1MelanomaNF-κB nuclear factor kappa BMTT 3-[45-dimethyltiazol-2-yl]-25-diphenyl tetrazolium bromideMelanomaNF-kappa BOpuntiaComplementary and Alternative Medicine2708 DermatologyBetaxanthinsCXCL1030220 oncology & carcinogenesisMolecular MedicinePhC phytochemicalGrowth inhibitionIndicaxanthinHumanBiologyPhytochemicalNHEM normal human epidermal melanocyte03 medical and health sciencesc-FLIP FLICE-inhibitory proteinIn vivoCell Line TumormedicineAnimalsHumansNeoplasm InvasivenessSkin NeoplasmCell ProliferationNeoplasm InvasiveneInflammationPharmacologyCell growthAnimalDrug Discovery3003 Pharmaceutical ScienceApoptosimedicine.diseaseMice Inbred C57BL030104 developmental biologyComplementary and alternative medicinechemistryTumor progressionList of Abbrevations: AxV-FITC annexin V-fluorescein isothiocyanateBetaxanthinFruitCutaneous melanomaCancer researchPI propidium iodide PIPhytomedicine : international journal of phytotherapy and phytopharmacology
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The effect of incorporating different concentrations of chlorhexidine digluconate on the degree of conversion of an experimental adhesive resin

2018

Background The aim of this study was to evaluate the effect of chlorhexidine digluconate incorporation on the degree of conversion of an experimental adhesive resin. Material and Methods The experimental resin was prepared from 70 wt% bisphenol A glycerolate dimethacrylate, 30 wt% hydroxyethyl methacrylate, silanized SiO2 nanofillers, 0.5% of camphorquinone and ethyl 4-dimethylaminebenzoate (binary photo-initiator system). Five chlorhexidine digluconate concentrations (0, 0.5, 1, 2 and 4 wt%) were then incorporated into the experimental resin. Thirty Potassium Bromide pellets were prepared then divided into six groups (n=5/group), repre¬senting the tested adhesive resins (Single Bond 2, 0, …

0301 basic medicineBisphenol AChemistryPotassium bromideResearchChlorhexidinePellets030206 dentistry(Hydroxyethyl)methacrylate:CIENCIAS MÉDICAS [UNESCO]Operative Dentistry and Endodontics03 medical and health scienceschemistry.chemical_compound030104 developmental biology0302 clinical medicinePolymerizationUNESCO::CIENCIAS MÉDICASmedicineAdhesiveFourier transform infrared spectroscopyGeneral DentistryNuclear chemistrymedicine.drug
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Enhanced autophagic-lysosomal activity and increased BAG3-mediated selective macroautophagy as adaptive response of neuronal cells to chronic oxidati…

2019

Oxidative stress and a disturbed cellular protein homeostasis (proteostasis) belong to the most important hallmarks of aging and of neurodegenerative disorders. The proteasomal and autophagic-lysosomal degradation pathways are key measures to maintain proteostasis. Here, we report that hippocampal cells selected for full adaptation and resistance to oxidative stress induced by hydrogen peroxide (oxidative stress-resistant cells, OxSR cells) showed a massive increase in the expression of components of the cellular autophagic-lysosomal network and a significantly higher overall autophagic activity. A comparative expression analysis revealed that distinct key regulators of autophagy are upregu…

0301 basic medicineClinical BiochemistryLFQ Label-free quantificationLETM Leucine zipper and EF-hand containing transmembrane proteinmedicine.disease_causeBiochemistryCHX Cycloheximide0302 clinical medicineBNIP3 Bcl-2 interacting protein 3RAPA RapamycinPIK3C3 Class III PI3‐kinasePhosphorylationlcsh:QH301-705.5Neuronslcsh:R5-920PolyUB PolyubiquitinChemistryBAG3OPA1 Optic atrophy 1TOR Serine-Threonine KinasesWIPI1 WD repeat domain phosphoinositide-interacting protein 1ATG Autophagy relatedTFEB Transcription factor EBCell biologyMitochondriasiRNA Small interfering RNADLP1 Dynamin-like protein 1LAMP1 Lysosomal‐associated membrane protein 1PURO Puromycinlcsh:Medicine (General)Protein homeostasisResearch PaperBafA1 Bafilomycin A1LAMP2 Lysosomal‐associated membrane protein 2Proteasome Endopeptidase ComplexRAB18 Member RAS oncogeneTUB TubulinLC3 Light chain 3 proteinOxidative phosphorylationBAG3CTSD Cathepsin DModels BiologicalCell Line03 medical and health sciencesDownregulation and upregulationMacroautophagymedicineAutophagyHumansAdaptationBAG1 Bcl-2-associated athanogene 1BECN1 Beclin1PI3K/AKT/mTOR pathwayAdaptor Proteins Signal TransducingTEM Transmission electron microscopyHsp70 Heat shock protein 70Organic ChemistryAutophagyAutophagosomesmTOR Mammalian target of rapamycinHsp70Oxidative Stress030104 developmental biologyProteostasislcsh:Biology (General)CV CanavanineBAG3 Bcl-2-associated athanogene 3MTT (3-(45-Dimethylthiazol-2-yl)-25-Diphenyltetrazolium Bromide)Apoptosis Regulatory ProteinsLysosomes030217 neurology & neurosurgeryOxidative stressRedox Biology
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FRET-based method for evaluation of the efficiency of reversible and irreversible sonoporation.

2017

It is widely known that not all of the treated cells survive after introduction of exogenous molecules via any physical method. Therefore, it is important to develop methods that would allow simultaneous evaluation of both molecular delivery efficiency and cell viability. This study presents Forster resonance energy transfer (FRET)-based method that allows molecular transfer and cell viability evaluation in a single measurement by employing two common fluorescent dyes, namely, ethidium bromide and trypan blue. The method has been validated using cell sonoporation. The FRET-based method allows the efficiency evaluation of both reversible and irreversible sonoporation in a single experiment. …

0301 basic medicineMaterials scienceCell SurvivalSonicationSingle measurementBiomedical EngineeringCHO CellsBiomaterials03 medical and health scienceschemistry.chemical_compoundSonicationCricetulusEthidiumFluorescence Resonance Energy TransferAnimalsHumansViability assayFluorescent DyesTrypan BlueFluorescenceAtomic and Molecular Physics and OpticsElectronic Optical and Magnetic Materials030104 developmental biologyFörster resonance energy transferchemistryBiophysicsTrypan blueEthidium bromideSonoporationJournal of biomedical optics
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CCDC 817434: Experimental Crystal Structure Determination

2011

Related Article: M.Giese, M.Albrecht, C.Bannwarth, G.Raabe, A.Valkonen, K.Rissanen|2011|Chem.Commun.|47|8542|doi:10.1039/c1cc12667a

1-(26-Difluorobenzyl)-4-aza-1-azoniabicyclo[2.2.2]octane bromide monohydrateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 177642: Experimental Crystal Structure Determination

2002

Related Article: M.I.Burguete, M.Bolte, J.C.Frias, E.Garcia-Espana, S.V.Luis, J.F.Miravet|2002|Tetrahedron|58|4179|doi:10.1016/S0040-4020(02)00381-2

26610-Tetrabenzyl-210-diaza-6-azonia(11)paracyclophane bromide chloroform solvateSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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CCDC 745351: Experimental Crystal Structure Determination

2011

Related Article: M.Albrecht, M.Muller, A.Valkonen, K.Rissanen|2010|CrystEngComm|12|3698|doi:10.1039/c003636f

4-Bromo-N-(pentafluorobenzyl)anilinium bromideSpace GroupCrystallographyCrystal SystemCrystal StructureCell ParametersExperimental 3D Coordinates
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FTIR quantitative analysis of calcium carbonate (calcite) and silica (quartz) mixtures using the constant ratio method. Application to geological sam…

2002

A methodology for quantifying calcium carbonate (875 and 712 cm(-1)) and silica (798 and 779 cm(-1)) by FTIR spectroscopy applying the constant ratio method is proposed. The studied method is applied for quantitative analysis of calcite and quartz in geological samples. The suggested method uses potassium ferricyanide (2115 cm(-1)) as standard and samples are prepared as potassium bromide pellets, with statistically satisfactory results (relative standard deviation less than 5%). The influence of particle size (pulverised samples) on the accuracy of the results found by FTIR spectroscopy applying the constant ratio method has been studied. The granulometric study suggests that the homogenei…

Absorbancechemistry.chemical_compoundCalcium carbonatechemistryPotassium bromidePelletsAnalytical chemistryCarbonateInfrared spectroscopyParticle sizeFourier transform infrared spectroscopyAnalytical ChemistryTalanta
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Functional Profile Of Aclidinium Bromide In Isolated Human Bronchi And Left Atria

2011

Aclidinium bromidebusiness.industryMedicinePharmacologybusinessA45. BRONCHODILATORS FOR COPD: OLD FAITHFULS AND NOVEL COMPOUNDS
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